TargetMol

LY2794193

Product Code:
 
TAR-T15807
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15807-5mg5mg£438.00
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TAR-T15807-50mg50mg£1,966.00
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Quantity:
TAR-T15807-100mg100mg£2,697.00
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This product comes from: United States.
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Further Information

Bioactivity:
LY2794193 is a highly effective and selective agonist of the mGlu3 receptor (hmGlu3 Ki=0.927 nM,EC50=0.47 nM; hmGlu2 Ki=412 nM,EC50=47.5 nM).
CAS:
2173037-97-1
Formula:
C16H18N2O6
Molecular Weight:
334.328
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
[H][C@]12[C@H](C(O)=O)[C@@]1([H])[C@@](N)(C[C@@H]2NC(=O)c1cccc(OC)c1)C(O)=O
Target:
SGLT

References

1. Monn JA, et al. Synthesis and Pharmacological Characterization of C4?-Amide-Substituted 2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylates. Identification of (1 S,2 S,4 S,5 R,6 S)-2-Amino-4-[(3-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid (LY2794193), a Highly Potent and Selective mGlu3 Receptor Agonist. J Med Chem. 2018 Mar 22;61(6):2303-2328.