TargetMol

PKI-166

Product Code:
 
TAR-T16549
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T16549-1mg1mg£189.00
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Quantity:
TAR-T16549-1mL1 mL * 10 mM (in DMSO)£287.00
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TAR-T16549-5mg5mg£369.00
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TAR-T16549-10mg10mg£517.00
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TAR-T16549-25mg25mg£790.00
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Quantity:
TAR-T16549-50mg50mg£1,050.00
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Quantity:
TAR-T16549-100mg100mg£1,396.00
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Quantity:
TAR-T16549-500mg500mg£2,713.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PKI-166 is an effective and selective EGFR tyrosine kinase inhibitor (IC50: 0.7 nM).
CAS:
187724-61-4
Formula:
C20H18N4O
Molecular Weight:
330.38
Pathway:
Tyrosine Kinase/Adaptors|Angiogenesis
Purity:
0.98
SMILES:
OC1=CC=C(C2=CC3=C(N=CN=C3N2)N[C@@H](C4=CC=CC=C4)C)C=C1
Target:
VEGFR

References

1. Bruns CJ, et al. Blockade of the epidermal growth factor receptor signaling by a novel tyrosine kinase inhibitor leads to apoptosis of endothelial cells and therapy of human pancreatic carcinoma. Cancer Res. 2000 Jun 1;60(11):2926-35.