TargetMol

VU0467485

Product Code:
 
TAR-T17245
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T17245-100mg100mgEnquire
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TAR-T17245-50mg50mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
VU0467485 is a potent and selective muscarinic acetylcholine receptor 4 positive allosteric modulator. VU0467485 potentiates the activity of ACh at M4 (EC50s: 26.6 nM and 78.8 nM at the rat and human M4 receptors, respectively). VU0467485 displays selectivity for M4 over human and rat M1/2/3/5.
CAS:
1451994-10-7
Formula:
C17H17FN4O2S
Molecular Weight:
360.41
Purity:
0.98
SMILES:
COc1ccc(CNC(=O)c2sc3nnc(C)c(C)c3c2N)cc1F