TargetMol

Amauromine

Product Code:
 
TAR-T36566
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T36566-5mg5mg£1,171.00
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Quantity:
TAR-T36566-50mg50mg£2,303.00
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Quantity:
TAR-T36566-100mg100mg£3,042.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 μM. It is also an antagonist of GPR18 (IC50 = 3.74 μM). Amauromine has vasodilatory activity.
CAS:
88360-87-6
Formula:
C32H36N4O2
Molecular Weight:
508.7
Purity:
0.98
SMILES:
C=CC(C)(C)[C@]1([C@@]2([H])NC3=C1C=CC=C3)C[C@]4([H])N2C([C@@](C[C@]5(C(C)(C)C=C)[C@@]6([H])NC7=C5C=CC=C7)([H])N6C4=O)=O