TargetMol

Glucagon Receptor Antagonist I

Product Code:
 
TAR-T37223
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T37223-5mg5mg£850.00
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Quantity:
TAR-T37223-50mg50mg£1,661.00
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Quantity:
TAR-T37223-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Glucagon receptor antagonist I is a competitive antagonist of the glucagon receptor (GCGR; IC50 = 181 nM). It blocks glucagon-induced glycogenolysis in primary human hepatocytes and isolated liver. Glucagon receptor antagonist I, at 50 mg/kg, reduces the increase in glucose levels observed after intraperitoneal administration of glucagon in humanized mice. Glucagon receptor antagonist inactive control does not prevent glucagon-mediated actions.
CAS:
438618-32-7
Formula:
C20H30N2OS
Molecular Weight:
346.5
Purity:
0.98
SMILES:
O=C(C(CC)CC)NC(S1)=C(C#N)C2=C1CC(C(C)(C)CC)CC2