TargetMol

XMU-MP-3

Product Code:
 
TAR-T39430
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T39430-10mg10mg£590.00
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Quantity:
TAR-T39430-50mg50mg£1,597.00
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Quantity:
TAR-T39430-100mg100mg£2,464.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
XMU-MP-3 is a potent non-covalent BTK inhibitor with IC 50 s of 10.7 nM and 17.0 nM for BTK WT and BTK C481S mutation in the presence of 10 μM ATP, respectively. XMU-MP-3 also induces apoptosis.
CAS:
2031152-08-4
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Fu Gui, et al. A Non-Covalent Inhibitor XMU-MP-3 Overrides Ibrutinib-Resistant Btk C481S Mutation in B-cell Malignancies. Br J Pharmacol. 2019 Dec;176(23):4491-4509.