TargetMol

Teneligliptin hydrobromide

Product Code:
 
TAR-T6999
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T6999-10mg10mg£103.00
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TAR-T6999-25mg25mg£121.00
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TAR-T6999-50mg50mg£161.00
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TAR-T6999-100mg100mg£217.00
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TAR-T6999-200mg200mg£303.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM.
CAS:
906093-29-6
Formula:
C44H65Br5N12O2S2
Molecular Weight:
1257.73
Pathway:
Proteases/Proteasome; Ubiquitination;
Purity:
1
SMILES:
Br.Br.Br.Br.Br.Cc1cc(N2CCN(CC2)[C@@H]2CN[C@@H](C2)C(=O)N2CCSC2)n(n1)-c1ccccc1.Cc1cc(N2CCN(CC2)[C@@H]2CN[C@@H](C2)C(=O)N2CCSC2)n(n1)-c1ccccc1
Target:
Proteasome; DPP-4

References

Ideta T, et al. Int J Mol Sci. 16(12):29207-18. Kishimoto M, et al. Diabetes Metab Syndr Obes. 2013, 6:187-95. Pujadas G, et al. Endocrine. 2016, [Epub ahead of print]. Sameshima A, et al. J Endocrinol. 2015, 227(1):25-36.