TargetMol

Vanoxerine dihydrochloride

Product Code:
 
TAR-T7153
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T7153-10mg10mg£113.00
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Quantity:
TAR-T7153-1mL1 mL * 10 mM (in DMSO)£117.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T7153-50mg50mg£214.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Vanoxerine dihydrochloride is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)
CAS:
67469-78-7
Formula:
C28H34Cl2F2N2O
Molecular Weight:
523.49
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
Cl.Cl.Fc1ccc(cc1)C(OCCN1CCN(CCCc2ccccc2)CC1)c1ccc(F)cc1
Target:
Dopamine Receptor

References

Contreras P C , Bremer M E , Rao T S . GBR-12909 and fluspirilene potently inhibited binding of [3H] (+)3-PPP to sigma receptors in rat brain[J]. Life Sciences, 1990, 47(22):PL133-7. Vanoxerine, a New Drug for Terminating Atrial Fibrillation and Flutter[J]. J Cardiovasc Electrophysiol, 2010, 21(3):311-319. Rothman R B , Baumann M H , Prisinzano T E , et al. Dopamine transport inhibitors based on GBR12909 and benztropine as potential medications to treat cocaine addiction[J]. Biochemical Pharmacology, 2008, 75(1):2-16.