TargetMol

[Leu5]-Enkephalin acetate(58822-25-6 free base)

Product Code:
 
TAR-T7173L
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7173L-10mg10mg£111.00
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TAR-T7173L-25mg25mg£152.00
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TAR-T7173L-50mg50mg£193.00
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TAR-T7173L-100mg100mg£255.00
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TAR-T7173L-200mg200mg£348.00
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Further Information

Bioactivity:
[Leu5]-Enkephalin acetate is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
CAS:
T7173L
Formula:
C28H37N5O7
Molecular Weight:
555.63
Pathway:
Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Purity:
0.9928
SMILES:
CC(O)=O.CC(C)C[C@@H](C(O)=O)NC([C@H](CC1=CC=CC=C1)NC(CNC(CNC([C@H](CC2=CC=C(O)C=C2)N)=O)=O)=O)=O
Target:
Opioid Receptor; Endogenous Metabolite

References

Meunier J C , Moisand C . Binding of leu5-enkephalin and met5-enkephalin to a particulate fraction from rat cerebrum[J]. Febs Letters, 1977, 77(2):0-213. Fabisiak A , Ma?gorzata Soboci?ska, El?bieta Kamysz, et al. Antinociceptive potency of enkephalins and enkephalinase inhibitors in the mouse model of colorectal distension - proof of concept[J]. Chemical Biology & Drug Design, 2018, 92(1).