TargetMol

IC87201

Product Code:
 
TAR-T7355
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7355-5mg5mg£124.00
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Quantity:
TAR-T7355-1mL1 mL * 10 mM (in DMSO)£140.00
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TAR-T7355-10mg10mg£155.00
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TAR-T7355-25mg25mg£254.00
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TAR-T7355-50mg50mg£346.00
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Quantity:
TAR-T7355-100mg100mg£470.00
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Further Information

Bioactivity:
IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.
CAS:
866927-10-8
Formula:
C13H10Cl2N4O
Molecular Weight:
309.15
Pathway:
Membrane transporter/Ion channel; Neuroscience;
Purity:
0.9744
SMILES:
Oc1c(Cl)cc(Cl)cc1CNc1ccc2nn[nH]c2c1
Target:
iGluR

References

Lee W H , Xu Z , Ashpole N M , et al. Small molecule inhibitors of PSD95-nNOS protein?protein interactions as novel analgesics[J]. Neuropharmacology, 2015:S0028390815002282. Bach A , Pedersen S W , Dorr L A , et al. Biochemical investigations of the mechanism of action of small molecules ZL006 and IC87201 as potential inhibitors of the nNOS-PDZ/PSD-95-PDZ interactions[J]. Scientific Reports, 2015, 5:12157.