TargetMol

[Leu5]-Enkephalin TFA(58822-25-6(free bas))

Product Code:
 
TAR-T7665
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7665-10mg10mg£108.00
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Quantity:
TAR-T7665-1mL1 mL * 10 mM (in DMSO)£128.00
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TAR-T7665-25mg25mg£149.00
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TAR-T7665-50mg50mg£189.00
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Quantity:
TAR-T7665-100mg100mg£249.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
[Leu5]-Enkephalin is the most potent δ-receptor ago
CAS:
73563-78-7
Formula:
C30H38F3N5O9
Molecular Weight:
669.655
Pathway:
Neuroscience; GPCR/G Protein; Metabolism; Endocrinology/Hormones
Purity:
0.9963
SMILES:
OC(=O)C(F)(F)F.CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(O)=O
Target:
Opioid Receptor; Endogenous Metabolite

References

Robert J Cassell , Krishna K Sharma , Hongyu Su,et al.The Meta-Position of Phe 4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors[J].Molecules, 24 (24) 2019 Dec 1 Meunier J C , Moisand C . Binding of leu5-enkephalin and met5-enkephalin to a particulate fraction from rat cerebrum[J]. Febs Letters, 1977, 77(2):0-213.