TargetMol

CGP 37849

Product Code:
 
TAR-T7720
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7720-1mg1mg£201.00
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TAR-T7720-5mg5mg£369.00
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TAR-T7720-10mg10mg£517.00
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TAR-T7720-25mg25mg£790.00
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TAR-T7720-50mg50mg£1,050.00
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Quantity:
TAR-T7720-100mg100mg£1,396.00
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This product comes from: United States.
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Further Information

Bioactivity:
CGP37849 is an effective and competitive NMDA receptor antagonist (Ki = 35 nM). CGP37849 is an anticonvulsive following oral administration in vivo.
CAS:
127910-31-0
Formula:
C6H12NO5P
Molecular Weight:
209.138
Pathway:
Neuroscience|Membrane transporter/Ion channel
Purity:
0.98
SMILES:
CC(CP(O)(O)=O)=C/C(N)C(O)=O
Target:
iGluR|NMDAR

References

Papp M, et al. Antidepressant activity of non-competitive and competitive NMDA receptor antagonists in a chronic mild stress model of depression. Eur J Pharmacol. 1994;263(1-2):1-7. Schmutz M, et al. The competitive NMDA receptor antagonists CGP 37849 and CGP 39551 are potent, orally-active anticonvulsants in rodents. Naunyn Schmiedebergs Arch Pharmacol. 1990;342(1):61-66. Przegali?ski E, et al. The influence of the benzodiazepine receptor antagonist flumazenil on the anxiolytic-like effects of CGP 37849 and ACPC in rats. Neuropharmacology. 2000;39(10):1858-1864. Fagg GE, et al. CGP 37849 and CGP 39551: novel and potent competitive N-methyl-D-aspartate receptor antagonists with oral activity. Br J Pharmacol. 1990;99(4):791-797.