TargetMol

Diphylline

Product Code:
 
TAR-T0892
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T0892-50mg50mg£108.00
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TAR-T0892-100mg100mg£120.00
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TAR-T0892-1mL1 mL * 10 mM (in DMSO)£125.00
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TAR-T0892-500mg500mg£214.00
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This product comes from: United States.
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Further Information

Bioactivity:
Dyphylline is a xanthine derivative. Dyphilline exerts bronchodilator effects and to a lesser extent vasodilator and diuretic properties. Dyphilline probably acts as a competitive inhibitor of phosphodiesterase which leads to an increase in intracellular cAMP. This results in relaxation of bronchial smooth muscle and other smooth muscles. Dyphylline may also antagonize adenosinereceptors. Dyphylline is used in the treatment of acute bronchial asthma, chronic bronchitis and emphysema.
CAS:
479-18-5
Formula:
C10H14N4O4
Molecular Weight:
254.246
Pathway:
Metabolism; GPCR/G Protein; Neuroscience
Purity:
0.991
SMILES:
Cn1c2ncn(CC(O)CO)c2c(=O)n(C)c1=O
Target:
PDE; Adenosine Receptor

References

1. Schwabe U, et al. Naunyn Schmiedebergs Arch Pharmacol. 1985 Sep;330(3):212-21.