TargetMol

GSK-5498A

Product Code:
 
TAR-T11473
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11473-5mg5mg£351.00
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TAR-T11473-50mg50mg£1,099.00
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Quantity:
TAR-T11473-100mg100mg£1,629.00
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This product comes from: United States.
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Further Information

Bioactivity:
GSK-5498A is a selective blocker of CARC (IC50, 1 μM). It inhibits mediator release from mast cells, and pro-inflammatory cytokine release from T-cells in a variety of species.
CAS:
1253186-49-0
Formula:
C18H11F6N3O
Molecular Weight:
399.296
Purity:
0.98
SMILES:
Fc1cccc(c1Cn1ccc(NC(=O)c2c(F)cccc2F)n1)C(F)(F)F

References

1. Rice LV, et al. Characterization of selective Calcium-Release Activated Calcium channel blockers in mast cells and T-cells from human, rat, mouse and guinea-pig preparations. Eur J Pharmacol. 2013 Mar 15;704(1-3):49-57.