TargetMol

LDN-192960 hydrochloride

Product Code:
 
TAR-T11830
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T11830-5mg5mg£264.00
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TAR-T11830-50mg50mg£870.00
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Quantity:
TAR-T11830-100mg100mg£1,283.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
LDN-192960 hydrochloride is an inhibitor of Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) and Haspin with IC50s of 48 nM and 10 nM, respectively.
CAS:
2309172-48-1
Formula:
C18H22Cl2N2O2S
Molecular Weight:
401.35
Purity:
0.98
SMILES:
NCCCSC1=C(C=C(OC)C=C2)C2=NC3=CC=C(OC)C=C31.Cl.Cl

References

1. Cuny GD, et al. Structure-activity relationship study of acridine analogs as haspin and DYRK2 kinase inhibitors. Bioorg Med Chem Lett. 2010 Jun 15;20(12):3491-4.