TargetMol

Nav1.7-IN-3

Product Code:
 
TAR-T12183
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12183-5mg5mg£337.00
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Quantity:
TAR-T12183-50mg50mg£1,532.00
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Quantity:
TAR-T12183-100mg100mg£2,319.00
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This product comes from: United States.
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Further Information

Bioactivity:
Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM).
CAS:
1788872-06-9
Formula:
C17H20ClFN4O2S2
Molecular Weight:
430.94
Purity:
0.98
SMILES:
Fc1cc(NCC23CCCN2CCC3)c(Cl)cc1S(=O)(=O)Nc1nccs1

References

1. Roecker AJ, et al. Discovery of selective, orally bioavailable, N-linked arylsulfonamide Nav1.7 inhibitors with pain efficacy in mice. Bioorg Med Chem Lett. 2017 May 15;27(10):2087-2093.