TargetMol

TrkA-IN-1

Product Code:
 
TAR-T13208
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13208-5mg5mg£304.00
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Quantity:
TAR-T13208-50mg50mg£1,219.00
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Quantity:
TAR-T13208-100mg100mg£1,813.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TrkA-IN-1 is a potent and selective inhibitor of Tropomyosin-related kinase A (TrkA) (IC50: 99 nM in a cell-based assay) with analgesic activity.
CAS:
1680179-43-4
Formula:
C25H20N4O
Molecular Weight:
392.462
Pathway:
Tyrosine Kinase/Adaptors
Purity:
0.98
SMILES:
Cc1ncc(NC(=O)NC2c3ccccc3-c3ccccc23)c(n1)-c1ccccc1
Target:
Trk receptor

References

1. Su HP , et al. Structural characterization of nonactive site, TrkA-selective kinase inhibitors. Proc Natl Acad Sci U S A. 2017 Jan 17;114(3):E297-E306.