TargetMol

Cyamemazine

Product Code:
 
TAR-T15026
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15026-50mg50mg£668.00
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TAR-T15026-100mg100mg£970.00
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Further Information

Bioactivity:
Cyamemazine, contains the phenothiazine chromophore, is a neuroleptic agent used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki: 12 nM), 5-HT2A (Ki: 1.5 nM) and 5-HT2C (Ki: 75 nM) receptors antagonist with antipsychotic activity.
CAS:
3546-03-0
Formula:
C19H21N3S
Molecular Weight:
323.46
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
CC(CN(C)C)CN1c2ccccc2Sc2ccc(cc12)C#N
Target:
5-HT Receptor

References

1. Bourin M, et al. Preclinical and clinical pharmacology of cyamemazine: anxiolytic effects and prevention of alcohol and benzodiazepine withdrawal syndrome. CNS Drug Rev. 2004 Fall;10(3):219-29. 2. Vendrell-Criado V, et al. Photobehavior of the antipsychotic drug cyamemazine in a supramolecular gel protective environment. J Photochem Photobiol B. 2020 Jan;202:111686.