TargetMol

Fosnetupitant

Product Code:
 
TAR-T15341
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15341-5mg5mg£850.00
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TAR-T15341-50mg50mg£1,661.00
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Quantity:
TAR-T15341-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.
CAS:
1703748-89-3
Formula:
C31H35F6N4O5P
Molecular Weight:
688.608
Purity:
0.98
SMILES:
CN(C(=O)C(C)(C)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cnc(cc1-c1ccccc1C)N1CC[N+](C)(COP(O)([O-])=O)CC1

References

1. Ruzza C, et al. In vitro and in vivo pharmacological characterization of Pronetupitant, a prodrug of the neurokinin 1 receptor antagonist Netupitant. Peptides. 2015 Jul;69:26-32.