TargetMol

Mivotilate

Product Code:
 
TAR-T16082
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16082-5mg5mg£270.00
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TAR-T16082-50mg50mg£1,026.00
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Quantity:
TAR-T16082-100mg100mg£1,564.00
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This product comes from: United States.
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Further Information

Bioactivity:
Mivotilate is a nontoxic, potent activator of the aryl hydrocarbon receptor (AhR). It acts as a hepatoprotective agent.
CAS:
130112-42-4
Formula:
C12H14N2O3S3
Molecular Weight:
330.44
Purity:
0.98
SMILES:
CC(C)OC(=O)C(C(=O)Nc1nc(C)cs1)=C1SCS1

References

1. Whelan F, et al. Amino acid substitutions in the aryl hydrocarbon receptor ligand binding domain reveal YH439 as an atypical AhR activator. Mol Pharmacol. 2010 Jun;77(6):1037-46. 2. Jeong KS, et al. Transcriptional inhibition of cytochrome P4502E1 by a synthetic compound, YH439. Arch Biochem Biophys. 1996 Feb 1;326(1):137-44. 3. Lee IJ, et al. Transcriptional induction of the cytochrome P4501A1 gene by a thiazolium compound, YH439. Mol Pharmacol. 1996 Jun;49(6):980-8.