TargetMol

Ro15-4513

Product Code:
 
TAR-T16775
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16775-5mg5mg£291.00
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TAR-T16775-50mg50mg£1,010.00
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TAR-T16775-100mg100mg£1,492.00
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Further Information

Bioactivity:
Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.
CAS:
91917-65-6
Formula:
C15H14N6O3
Molecular Weight:
326.316
Purity:
0.98
SMILES:
CCOC(=O)c1ncn-2c1CN(C)C(=O)c1cc(ccc-21)N=[N+]=[N-]

References

1. Bonetti EP, et al. Ro 15-4513: partial inverse agonism at the BZR and interaction with ethanol. Pharmacol Biochem Behav. 1988 Nov;31(3):733-49. 2. Suzdak PD, et al. Effects of Ro15-4513 and other benzodiazepine receptor inverse agonists on alcohol-inducedintoxication in the rat. J Pharmacol Exp Ther. 1988 Jun;245(3):880-6. 3. Linden AM, et al. Ro 15-4513 Antagonizes Alcohol-Induced Sedation in Mice Through ???2-type GABA(A) Receptors. Front Neurosci. 2011 Jan 20;5:3.