TargetMol

RPR-260243

Product Code:
 
TAR-T16796
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16796-5mg5mg£343.00
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TAR-T16796-50mg50mg£1,187.00
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Quantity:
TAR-T16796-100mg100mg£1,749.00
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Further Information

Bioactivity:
RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM).
CAS:
668463-35-2
Formula:
C28H25F3N2O4
Molecular Weight:
510.5
Purity:
0.98
SMILES:
O=C([C@H]1CN(CC#CC2=CC(F)=CC(F)=C2F)CC[C@H]1CCC(C3=CC=NC4=CC=C(OC)C=C34)=O)O

References

1. Kang J, et al. Discovery of a small molecule activator of the human ether-a-go-go-related gene (HERG) cardiac K+ channel. Mol Pharmacol. 2005 Mar;67(3):827-36.