TargetMol

GLPG0492

Product Code:
 
TAR-T11410L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T11410L-1mg1mg£182.00
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TAR-T11410L-2mg2mg£229.00
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TAR-T11410L-5mg5mg£349.00
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TAR-T11410L-1mL1 mL * 10 mM (in DMSO)£377.00
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TAR-T11410L-10mg10mg£470.00
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TAR-T11410L-25mg25mg£707.00
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TAR-T11410L-50mg50mg£978.00
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TAR-T11410L-100mg100mg£1,291.00
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This product comes from: United States.
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Further Information

Bioactivity:
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic activity on the prostate.
CAS:
1215085-92-9
Formula:
C19H14F3N3O3
Molecular Weight:
389.334
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
CN1C(=O)N(C(=O)[C@@]1(CO)c1ccccc1)c1ccc(C#N)c(c1)C(F)(F)F
Target:
Androgen Receptor

References

Nique F, et al. Identification of a 4-(hydroxymethyl)diarylhydantoin as a selective androgen receptor modulator. J Med Chem. 2012 Oct 11;55(19):8236-47. Cozzoli A, et al. GLPG0492, a novel selective androgen receptor modulator, improves muscle performance in the exercised-mdx mouse model of muscular dystrophy. Pharmacol Res. 2013 Jun;72:9-24. Blanqu? R, et al. Characterization of GLPG0492, a selective androgen receptor modulator, in a mouse model of hindlimb immobilization. BMC Musculoskelet Disord. 2014 Sep 3;15:291.