TargetMol

THZ1-R

Product Code:
 
TAR-T13153
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T13153-5mg5mg£378.00
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Quantity:
TAR-T13153-50mg50mg£1,508.00
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Quantity:
TAR-T13153-100mg100mg£2,095.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
THZ1-R displays diminished activity for CDK7 inhibition(Kd:142 nM).
CAS:
1621523-07-6
Formula:
C31H30ClN7O2
Molecular Weight:
568.08
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
CN(C)CCCC(=O)Nc1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(Cl)c(n2)-c2c[nH]c3ccccc23)c1
Target:
CDK

References

1. Kwiatkowski N, et al. Targeting transcription regulation in cancer with a covalent CDK7 inhibitor. Nature. 2014 Jul 31;511(7511):616-20.