TargetMol

TP-004

Product Code:
 
TAR-T13188
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T13188-5mg5mg£337.00
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Quantity:
TAR-T13188-50mg50mg£1,332.00
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Quantity:
TAR-T13188-100mg100mg£2,070.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TP-004 is a potent and reversible methionine aminopeptidase 2 (MetAP2) inhibitor (IC50: 6 nM).
CAS:
1454299-21-8
Formula:
C17H16F3N5O
Molecular Weight:
363.344
Purity:
0.98
SMILES:
Cc1nc(ncc1-c1cc(cc2[nH]ncc12)C(F)(F)F)N1CC[C@@H](O)C1

References

1. Cheruvallath, Z., et al. Discovery of potent, reversible MetAP2 inhibitors via fragment based drug discovery and structure based drug design?Part Bioorganic & Medicinal Chemistry Letters, 26(12), 2774?2778.