TargetMol

Vofopitant dihydrochloride

Product Code:
 
TAR-T13329L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T13329L-5mg5mg£302.00
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TAR-T13329L-50mg50mg£1,163.00
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Quantity:
TAR-T13329L-100mg100mg£1,564.00
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This product comes from: United States.
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Further Information

Bioactivity:
Vofopitant dihydrochloride is a selective and orally available antagonist of tachykinin neurokinin 1(NK1) receptor (pKi: 9.5 and 10.6 in rat and human membranes respectively) and is a potential broad-spectrum anti-emetic agent.
CAS:
168266-51-1
Formula:
C21H25Cl2F3N6O
Molecular Weight:
505.37
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
Cl.Cl.COc1ccc(cc1CN[C@H]1CCCN[C@H]1c1ccccc1)-n1nnnc1C(F)(F)F
Target:
Neurokinin receptor

References

1. Gardner CJ, et al. GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity. Regul Pept. 1996 Aug 27;65(1):45-53.