TargetMol

BMS-193885

Product Code:
 
TAR-T14671
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14671-1mg1mg£109.00
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TAR-T14671-5mg5mg£168.00
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TAR-T14671-1mL1 mL * 10 mM (in DMSO)£198.00
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TAR-T14671-10mg10mg£229.00
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TAR-T14671-25mg25mg£389.00
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TAR-T14671-50mg50mg£544.00
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TAR-T14671-100mg100mg£748.00
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Further Information

Bioactivity:
BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a Ki of 3.3 nM, and an IC50 of 5.9 nM for hY1.
CAS:
186185-03-5
Formula:
C33H42N4O6
Molecular Weight:
590.71
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
O=C(OC)C1=C(NC(=C(C(=O)OC)C1C=2C=CC=C(C2)NC(=O)NCCCN3CCC(C=4C=CC=C(OC)C4)CC3)C)C
Target:
Neuropeptide Y Receptor

References

Poindexter GS, et al. Dihydropyridine neuropeptide Y Y(1) receptor antagonists. Bioorg Med Chem Lett. 2002 Feb 11;12(3):379-82. Antal-Zimanyi I, et al. Pharmacological characterization and appetite suppressive properties of BMS-193885, a novel and selective neuropeptide Y(1) receptor antagonist. Eur J Pharmacol. 2008 Aug 20;590(1-3):224-32.