TargetMol

DC_517

Product Code:
 
TAR-T15081
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15081-5mg5mg£351.00
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TAR-T15081-50mg50mg£1,508.00
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Quantity:
TAR-T15081-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
DC_517 is an inhibitor of DNA methyltransferase 1 (DNMT1) ( IC50: 1.7 μM; Kd: 0.91 μM).
CAS:
500017-70-9
Formula:
C33H35N3O2
Molecular Weight:
505.662
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
CC(C)NCC(O)COC(Cn1c2ccccc2c2ccccc12)Cn1c2ccccc2c2ccccc12
Target:
DNA Methyltransferase

References

1. Chen S, et al. Identifying novel selective non-nucleoside DNA methyltransferase 1 inhibitors through docking-based virtual screening. J Med Chem. 2014 Nov 13;57(21):9028-9041.