TargetMol

PSI-697

Product Code:
 
TAR-T16676
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16676-5mg5mg£1,010.00
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TAR-T16676-50mg50mg£1,982.00
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TAR-T16676-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
PSI-697 is an inhibitor of oral P-selectin (IC50: 125 μM).
CAS:
851546-61-7
Formula:
C21H18ClNO3
Molecular Weight:
367.83
Purity:
0.98
SMILES:
OC(=O)c1c(O)c(Cc2ccc(Cl)cc2)nc2c3CCCCc3ccc12

References

1. Bedard PW et al. Characterization of the novel P-selectin inhibitor PSI-697 [2-(4-chlorobenzyl)-3-hydroxy-7,8,9,10-tetrahydrobenzo[h] quinoline-4-carboxylic acid] in vitro and in rodent models of vascular inflammation and thrombosis. J Pharmacol Exp Ther. 2. Myers DD Jr et al. Resolution of venous thrombosis using a novel oral small-molecule inhibitor of P-selectin (PSI-697) without anticoagulation. Thromb Haemost. 2007 Mar;97(3):400-7. 3. Myers DD Jr et al. Treatment with an oral small molecule inhibitor of P selectin (PSI-697) decreases vein wall injury in a rat stenosis model of venous thrombosis. J Vasc Surg. 2006 Sep;44(3):625-32.