TargetMol

Flesinoxan

Product Code:
 
TAR-T16711
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16711-5mg5mg£371.00
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TAR-T16711-50mg50mg£1,332.00
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Quantity:
TAR-T16711-100mg100mg£1,966.00
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This product comes from: United States.
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Further Information

Bioactivity:
Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).
CAS:
98206-10-1
Formula:
C22H26FN3O4
Molecular Weight:
415.465
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
OC[C@@H]1COc2c(O1)cccc2N1CCN(CCNC(=O)c2ccc(F)cc2)CC1
Target:
5-HT Receptor

References

1. Hadrava V, et al. Characterization of 5-hydroxytryptamine1A properties of flesinoxan: in vivo electrophysiology and hypothermia study. Neuropharmacology. 1995 Oct;34(10):1311-26. 2. Schoeffter P, et al. Centrally acting hypotensive agents with affinity for 5-HT1A binding sites inhibit forskolin-stimulated adenylate cyclase activity in calf hippocampus. Br J Pharmacol. 1988 Nov;95(3):975-85. 3. Rodgers RJ, et al. Antianxiety and behavioral suppressant actions of the novel 5-HT1A receptor agonist, flesinoxan. Pharmacol Biochem Behav. 1994 Aug;48(4):959-63.