TargetMol

Eplivanserin hemifumarate

Product Code:
 
TAR-T27277
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27277-50mg50mg£703.00
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Quantity:
TAR-T27277-100mg100mg£1,026.00
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This product comes from: United States.
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Further Information

Bioactivity:
Eplivanserin is an inverse agonist of 5-HT2A.
CAS:
130580-02-8
Formula:
C23H25FN2O6
Molecular Weight:
444.459
Purity:
0.98
SMILES:
OC(=O)C=CC(O)=O.CN(C)CCON=C(C=Cc1ccc(O)cc1)/c1ccccc1F

References

1. Heller HC, Salehi A, Chuluun B, Das D, Lin B, Moghadam S, Garner CC, Colas D. Nest building is impaired in the Ts65Dn mouse model of Down syndrome and rescued by blocking 5HT2a receptors. Neurobiol Learn Mem. 2014 Dec;116:162-71. doi: 10.1016/j.nlm.2014.10.002. Epub 2014 Oct 29. PubMed PMID: 25463650. 2. Dougherty JP, Oristaglio J. Chronic treatment with the serotonin 2A/2C receptor antagonist SR 46349B enhances the retention and efficiency of rule-guided behavior in mice. Neurobiol Learn Mem. 2013 Jul;103:50-63. doi: 10.1016/j.nlm.2013.04.002. Epub 2013 Apr 12. PubMed PMID: 23587729. 3. Griebel G, Beesk? S, Jacquet A, Laufrais C, Alonso R, Decobert M, Avenet P, Fran?on D. Further evidence for the sleep-promoting effects of 5-HT?A receptor antagonists and demonstration of synergistic effects with the hypnotic, zolpidem in rats. Neuropharmacology. 2013 Jul;70:19-26. doi: 10.1016/j.neuropharm.2012.12.008. Epub 2013 Jan 12. PubMed PMID: 23321054. 4. Ebdrup BH, Rasmussen H, Arnt J, Glenth?j B. Serotonin 2A receptor antagonists for treatment of schizophrenia. Expert Opin Investig Drugs. 2011 Sep;20(9):1211-23. doi: 10.1517/13543784.2011.601738. Epub 2011 Jul 8. Review. PubMed PMID: 21740279.