TargetMol

TASP0433864

Product Code:
 
TAR-T28928
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28928-5mg5mg£850.00
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TAR-T28928-50mg50mg£1,661.00
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Quantity:
TAR-T28928-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
TASP0433864 is a positive allosteric modulator of metabotropic glutamate 2 receptor with EC50 values of 199 and 206 nM at human and rat mGlu2 receptors, respectively, without exerting agonist activity at rat mGlu2 receptor.
CAS:
1431980-60-7
Formula:
C18H23N3O3
Molecular Weight:
329.4
Purity:
0.98
SMILES:
Cc1c(nc2O[C@H](COc3ccc(cc3)C(C)(C)C)Cn12)C(N)=O

References

1. Hiyoshi T, Marumo T, Hikichi H, Tomishima Y, Urabe H, Tamita T, Iida I, Yasuhara A, Karasawa J, Chaki S. Neurophysiologic and antipsychotic profiles of TASP0433864, a novel positive allosteric modulator of metabotropic glutamate 2 receptor. J Pharmacol Exp Ther. 2014 Dec;351(3):642-53. doi: 10.1124/jpet.114.218651. PubMed PMID: 25277141.