TargetMol

SAR 216471 hydrochloride

Product Code:
 
TAR-T36759
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T36759-5mg5mg£1,332.00
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TAR-T36759-50mg50mg£2,625.00
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Quantity:
TAR-T36759-100mg100mg£3,524.00
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This product comes from: United States.
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Further Information

Bioactivity:
Potent P2Y12 antagonist (IC50 = 17 nM). Displays antiplatelet and antithrombotic activity in vivo. Orally available.
CAS:
1279829-64-9
Formula:
C28H31ClN8O3.HCl
Molecular Weight:
599.51
Purity:
0.98
SMILES:
ClC1=CC=C2C(C(C(NC3=CC=C(N4C(C)=C(C(CCC)=O)C=N4)N=N3)=O)=CN2CC(N5CCN(C)CC5)=O)=C1.Cl

References

Boldron et al (2014) N-[6-(4-butanoyl-5-methyl-1H-pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1H-indole-3-carboxamide (SAR216471), a novel intravenous and oral, reversible, and directly acting P2Y12 antagonist. J.Med.Chem. 57 7293 PMID:25075638