TargetMol

SET 2

Product Code:
 
TAR-T37097
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T37097-1mg1mg£101.00
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Quantity:
TAR-T37097-5mg5mg£142.00
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Quantity:
TAR-T37097-1mL1 mL * 10 mM (in DMSO)£158.00
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Quantity:
TAR-T37097-10mg10mg£189.00
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Quantity:
TAR-T37097-25mg25mg£322.00
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Quantity:
TAR-T37097-50mg50mg£495.00
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Quantity:
TAR-T37097-100mg100mg£688.00
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Quantity:
TAR-T37097-500mg500mg£1,340.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TRPV2 (transient receptor potential vanilloid type 2) antagonist (IC50 = 0.46 μM). Selective for TRPV2 over TRPV1, TRPV3 and TRPV4 expressed in HEK293 cells. Inhibits lyosphosphatidic acid (LPA)-induced prostate cancer cell migration in vitro.
CAS:
2313525-20-9
Formula:
C17H21F3N4O2S
Molecular Weight:
402.44
Pathway:
Membrane transporter/Ion channel
Purity:
0.98
SMILES:
CCCN(C1=NC(SCCC(NCC2=CC=CO2)=O)=NC(C(F)(F)F)=C1)C
Target:
TRP/TRPV Channel

References

Chai H, et al. Structure-Based Discovery of a Subtype-Selective Inhibitor Targeting a Transient Receptor Potential Vanilloid Channel. J Med Chem. 2019 Feb 14;62(3):1373-1384.