TargetMol

Ethacizine hydrochloride

Product Code:
 
TAR-T11239
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
Ethacizine hydrochloride inhibits the depolarizing current responsible for the intraatrial and His-Purkinje-ventricular conduction. Ethacizine hydrochloride is a longer-lasting Class Ic antiarrhythmic agent than Flecainide.
CAS:
57530-40-2
Formula:
C22H28ClN3O3S
Molecular Weight:
449.99
Purity:
0.98
SMILES:
Cl.CCOC(=O)Nc1ccc2Sc3ccccc3N(C(=O)CCN(CC)CC)c2c1

References

1. Sugiyama A, et al. Comparison of cardiovascular effects of a novel class Ic antiarrhythmic agent, NIK-244, with those of flecainide in isolated canine heart preparations cross-circulated with a donor dog.Jpn J Pharmacol. 1991 May;56(1):1-12. 2. Satoh H, et al. An electrophysiological comparison of a novel class Ic antiarrhythmic agent, NIK-244 (ethacizin) and flecainide in canine ventricular muscle.Br J Pharmacol. 1989 Nov;98(3):827-32.Med Chem.?2019 Nov 6:115132.