TargetMol

GSK 4027

Product Code:
 
TAR-T11495L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T11495L-100mg100mgEnquire
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TAR-T11495L-50mg50mgEnquire
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Further Information

Bioactivity:
GSK 4027 is a PCAF/GCN5 bromodomain chemical probe. In a time-resolved fluorescence resonance energy transfer (TR-FRET) assay, it has a pIC50 of 7.4?0.11 for PCAF.
CAS:
2079896-25-4
Formula:
C17H21BrN4O
Molecular Weight:
377.286
Purity:
0.98
SMILES:
CN1C[C@@H](C[C@@H](C1)c1ccccc1)Nc1cnn(C)c(=O)c1Br

References

1. Humphreys PG, et al. Discovery of a Potent, Cell Penetrant, and Selective p300/CBP-Associated Factor (PCAF)/General Control Nonderepressible 5 (GCN5) Bromodomain Chemical Probe. J Med Chem. 2017 Jan 26;60(2):695-709.