TargetMol

SB 243213 hydrochloride

Product Code:
 
TAR-T12859
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12859-5mg5mg£1,251.00
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TAR-T12859-50mg50mg£2,464.00
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Quantity:
TAR-T12859-100mg100mg£3,283.00
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This product comes from: United States.
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Further Information

Bioactivity:
SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).It has improved anxiolytic profile and has the potential for schizophrenia and motor disorders.
CAS:
200940-23-4
Formula:
C22H20ClF3N4O2
Molecular Weight:
464.87
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
Cl.Cc1cc2CCN(C(=O)Nc3ccc(Oc4cccnc4C)nc3)c2cc1C(F)(F)F
Target:
5-HT Receptor

References

1. Wood MD, et al. SB-243213; a selective 5-HT2C receptor inverse agonist with improved anxiolytic profile: lack of tolerance and withdrawal anxiety. Neuropharmacology. 2001 Aug;41(2):186-99.