TargetMol

JNJ-46778212

Product Code:
 
TAR-T15619
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T15619-100mg100mgEnquire
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Further Information

Bioactivity:
JNJ-46778212 is an effective mGlu5 allosteric modulator (EC50: 260 nM).
CAS:
1363281-27-9
Formula:
C20H17FN2O3
Molecular Weight:
352.365
Pathway:
Neuroscience
Purity:
0.98
SMILES:
Fc1ccc(cc1)C(=O)N1CCc2nc(COc3ccccc3)oc2C1
Target:
GluR

References

1. Conde-Ceide S, et al. Discovery of VU0409551/JNJ-46778212: An mGlu5 Positive Allosteric Modulator Clinical Candidate Targeting Schizophrenia. ACS Med Chem Lett. 2015 May 20;6(6):716-20.