TargetMol

OGT 2115

Product Code:
 
TAR-T16380
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16380-1mg1mg£95.00
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TAR-T16380-5mg5mg£127.00
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TAR-T16380-1mL1 mL * 10 mM (in DMSO)£132.00
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TAR-T16380-10mg10mg£171.00
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TAR-T16380-25mg25mg£289.00
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TAR-T16380-50mg50mg£436.00
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TAR-T16380-100mg100mg£610.00
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This product comes from: United States.
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Further Information

Bioactivity:
OGT 2115 is an effective and cell-permeable heparanase inhibitor (IC50: 0.4 μM). OGT 2115 also suppresses heparan sulfate degradation activity. OGT 2115 has anti-angiogenic properties (IC50: 1 μM).
CAS:
853929-59-6
Formula:
C24H16BrFN2O4
Molecular Weight:
495.304
Purity:
0.98
SMILES:
OC(=O)Cc1ccc2oc(nc2c1)-c1ccc(NC(=O)C=Cc2ccc(Br)cc2)c(F)c1

References

1. Courtney SM, et al. Furanyl-1,3-thiazol-2-yl and benzoxazol-5-yl acetic acid derivatives: novel classes of heparanase inhibitor. Bioorg Med Chem Lett. 2005 May 2;15(9):2295-9. 2. Li Y, et al. Suppression of endoplasmic reticulum stress-induced invasion and migration of breast cancer cells through the downregulation of heparanase. Int J Mol Med. 2013 May;31(5):1234-42.