TargetMol

PD173212

Product Code:
 
TAR-T16448
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T16448-1mg1mg£124.00
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TAR-T16448-2mg2mg£148.00
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TAR-T16448-5mg5mg£213.00
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TAR-T16448-1mL1 mL * 10 mM (in DMSO)£258.00
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TAR-T16448-10mg10mg£281.00
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TAR-T16448-25mg25mg£426.00
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TAR-T16448-50mg50mg£586.00
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TAR-T16448-100mg100mg£780.00
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Quantity:
TAR-T16448-500mg500mg£1,500.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PD173212 is a selective N-type voltage-sensitive calcium channel (VSCC) blocker. It has an IC50 of 36 nM in IMR-32 assays.
CAS:
217171-01-2
Formula:
C38H53N3O3
Molecular Weight:
599.86
Pathway:
Membrane transporter/Ion channel|Metabolism
Purity:
0.98
SMILES:
CC(C)C[C@H](N(C)Cc1ccc(cc1)C(C)(C)C)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NC(C)(C)C
Target:
Calcium Channel

References

1. Hu LY, et al. Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers. Bioorg Med Chem Lett. 1999 Aug 2;9(15):2151-6.