TargetMol

Pumosetrag Hydrochloride

Product Code:
 
TAR-T16683
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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This product comes from: United States.
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Further Information

Bioactivity:
Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease.
CAS:
194093-42-0
Formula:
C15H18ClN3O2S
Molecular Weight:
339.84
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
Cl.O=C(N[C@H]1CN2CCC1CC2)c1c[nH]c2ccsc2c1=O
Target:
5-HT Receptor

References

1. Chetty N, et al. Effects of the novel 5-HT3 agonist MKC-733 on the rat, mouse and guinea pig digestive tract. Pharmacology. 2008;81(2):104-9. Epub 2007 Oct 19. 2. Coleman NS, et al. Effect of a novel 5-HT3 receptor agonist MKC-733 on upper gastrointestinal motility in humans. Aliment Pharmacol Ther. 2003 Nov 15;18(10):1039-48.