TargetMol

CPI-455 HCl

Product Code:
 
TAR-T22299
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T22299-5mg5mg£850.00
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Quantity:
TAR-T22299-50mg50mg£1,661.00
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Quantity:
TAR-T22299-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CPI-455 is a specific KDM5 inhibitor with IC50 value of 10 ? 1 nM for full-length KDM5A in enzymatic assays, elevating global levels of H3K4 trimethylation (H3K4me3) and decreased the number of DTPs in multiple cancer cell line models treated with targeted agents or standard chemotherapy.
CAS:
2095432-28-1
Formula:
C16H15ClN4O
Molecular Weight:
314.77
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
Cl.CC(C)c1c([nH]c2c(cnn2c1=O)C#N)-c1ccccc1
Target:
Histone Demethylase