TargetMol

(S)-Willardiine

Product Code:
 
TAR-T13456
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13456-5mg5mg£111.00
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TAR-T13456-10mg10mg£132.00
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TAR-T13456-50mg50mg£347.00
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Quantity:
TAR-T13456-100mg100mg£484.00
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This product comes from: United States.
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Further Information

Bioactivity:
(S)-Willardiine is a potent AMPA/kainate receptors agonist(EC50 : 44.8 uM).
CAS:
21416-43-3
Formula:
C7H9N3O4
Molecular Weight:
199.166
Pathway:
Membrane transporter/Ion channel|Neuroscience
Purity:
0.98
SMILES:
N[C@@H](Cn1ccc(=O)[nH]c1=O)C(O)=O
Target:
iGluR

References

1. Patneau DK, et al. Activation and desensitization of AMPA/kainate receptors by novel derivatives of willardiine. J Neurosci. 1992 Feb;12(2):595-606. 2. Fukushima T, et al. Calcium inhibits willardiine-induced responses in kainate receptor GluR6(Q)/KA-2. Neuroreport. 2001 Jan 22;12(1):163-7. 3. Gressens P, et al. The effects of AMPA receptor antagonists in models of stroke and neurodegeneration. Eur J Pharmacol. 2005 Sep 5;519(1-2):58-67.