TargetMol

AM-2099

Product Code:
 
TAR-T14201
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T14201-100mg100mgEnquire
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TAR-T14201-50mg50mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
AM-2099 is a voltage-gated sodium channel Nav1.7 inhibitor (IC50: 0.16 μM).
CAS:
1443373-17-8
Formula:
C19H13F3N4O3S2
Molecular Weight:
466.45
Purity:
0.98
SMILES:
COc1cc(ccc1-c1ncnc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F

References

1. Marx IE, et al. Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement. ACS Med Chem Lett. 2016 Sep 21;7(12):1062-1067.