TargetMol

Arachidonoyl 2'-Chloroethylamide

Product Code:
 
TAR-T38138
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38138-5mg5mg£850.00
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TAR-T38138-50mg50mg£1,661.00
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Quantity:
TAR-T38138-100mg100mg£2,079.00
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Further Information

Bioactivity:
Arachidonoyl 2-chloroethylamide (ACEA) is a potent and selective cannabinoid (CB) receptor 1 agonist with Ki values of 1.4 and >2,000 nM for CB1 and CB2 receptors, respectively. In whole animal experiments, ACEA induces hypothermia in mice with the same efficacy as arachidonoyl ethanolamide , in spite of its higher affinity for the CB1 receptor. These data have been interpreted to indicate that ACEA may be a substrate for fatty acid amide hydrolase (FAAH), and thus only transiently available in whole animal experiments.
CAS:
220556-69-4
Formula:
C22H36ClNO
Molecular Weight:
366
Purity:
0.98
SMILES:
CCCCC/C=CC/C=CC/C=CC/C=CCCCC(=O)NCCCl

References

Hillard, C.J., Manna, S., Greenberg, M.J., et al. Synthesis and characterization of potent and selective agonists of the neuronal cannabinoid receptor (CB1) J. Pharmacol. Exp. Ther. 289(3), 1427-1433 (1999). Pertwee, R.G. Pharmacology of cannabinoid receptor ligands Curr. Med. Chem. 6(8), 635-664 (1999).