TargetMol

Pimethixene maleate

Product Code:
 
TAR-T12489L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12489L-5mg5mg£96.00
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TAR-T12489L-50mg50mg£149.00
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TAR-T12489L-100mg100mg£203.00
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Further Information

Bioactivity:
Pimethixene maleate is a highly potent5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(with pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
CAS:
13187-06-9
Formula:
C23H23NO4S
Molecular Weight:
409.5
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
OC(=O)C=C/C(O)=O.CN1CCC(CC1)=C1c2ccccc2Sc2ccccc12
Target:
5-HT Receptor

References

1. Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80.