TargetMol

EPZ020411

Product Code:
 
TAR-T4314
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T4314-10mg10mgEnquire
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TAR-T4314-1mg1mgEnquire
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TAR-T4314-2mg2mgEnquire
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TAR-T4314-5mg5mgEnquire
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Further Information

Bioactivity:
EPZ020411 is a specific and effective inhibitor of PRMT6 (IC50=10 nM).
CAS:
1700663-41-7
Molecular Weight:
442.6
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
CNCCN(C)Cc1c[nH]nc1-c1ccc(O[C@H]2C[C@@H](C2)OCCC2CCOCC2)cc1
Target:
Histone Methyltransferase

References

Mitchell LH, et al. Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 ToolCompound. ACS Med Chem Lett. 2015 Apr 6;6(6):655-659.