TargetMol

MSC-4106

Product Code:
 
TAR-T60148
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T60148-1mg1mg£148.00
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TAR-T60148-5mg5mg£269.00
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TAR-T60148-1mL1 mL * 10 mM (in DMSO)£338.00
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TAR-T60148-10mg10mg£389.00
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TAR-T60148-25mg25mg£603.00
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TAR-T60148-50mg50mg£830.00
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Quantity:
TAR-T60148-100mg100mg£1,099.00
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This product comes from: United States.
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Further Information

Bioactivity:
MSC-4106 is an orally active and potent inhibitor of YAP/TAZ-TEAD. MSC-4106 inhibits TEAD1 or TEAD3 auto-palmitoylation and exhibits inhibitory effect on NCI-H226 tumor xenograft model [1].
CAS:
2738542-58-8
Molecular Weight:
359.3
Pathway:
Stem Cells
Purity:
1
SMILES:
O=C(O)C=1C=CC2=C(C1)C3=CN(N=C3N2C4=CC=C(C=C4)C(F)(F)F)C
Target:
YAP

References

Timo Heinrich, et al. Optimization of TEAD P-site binding fragment hit into in vivo active lead MSC-4106. J. Med. Chem. 2022, 65, 13, 9206?9229.