TargetMol

TUG-499

Product Code:
 
TAR-T60184
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T60184-1mg1mg£119.00
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TAR-T60184-5mg5mg£180.00
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TAR-T60184-1mL1 mL * 10 mM (in DMSO)£182.00
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TAR-T60184-10mg10mg£230.00
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TAR-T60184-25mg25mg£333.00
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TAR-T60184-50mg50mg£386.00
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TAR-T60184-100mg100mg£540.00
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TAR-T60184-500mg500mg£1,091.00
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This product comes from: United States.
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Further Information

Bioactivity:
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 has an affinity for FFAR1 or GPR40 over the related receptors FFA2, FFA3 and the nuclear receptor PPARγ, as well as other different receptors, ion channels and transporter proteins.TUG-499 can be used to study type 2 Type 2 diabetes.
CAS:
1206629-08-4
Molecular Weight:
320.17
Pathway:
DNA Damage/DNA Repair|Endocrinology/Hormones|Metabolism|GPCR/G Protein
Purity:
0.9959
SMILES:
O=C(O)CCC1=CC=C(C#CC=2C=C(Cl)N=C(Cl)C2)C=C1
Target:
GPR|PPAR

References

Christiansen E, et al. Identification of a potent and selective free fatty acid receptor 1 (FFA1/GPR40) agonist with favorable physicochemical and in vitro ADME properties. J Med Chem. 2011;54(19):6691-6703.