TargetMol

CDK9-IN-15

Product Code:
 
TAR-T60619
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T60619-1mg1mg£103.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T60619-1mL1 mL * 10 mM (in DMSO)£146.00
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Quantity:
TAR-T60619-5mg5mg£148.00
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Quantity:
TAR-T60619-10mg10mg£201.00
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Quantity:
TAR-T60619-25mg25mg£329.00
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Quantity:
TAR-T60619-50mg50mg£454.00
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Quantity:
TAR-T60619-100mg100mg£623.00
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Quantity:
TAR-T60619-500mg500mg£1,211.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
CDK9-IN-15 is a potent small molecule CDK9 inhibitor, which can block the phosphorylation of positive transcription elongation factor b (P-TEFb) on the C-terminal region of RNA Poly-II by degradation and inhibition of CDK9, inhibit transcription, and rapidly reduce the level of intracellular mRNA, thereby causing apoptosis of tumor cells.
CAS:
852678-17-2
Molecular Weight:
293.34
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
OC1=CC=CC=2C(=CC=CC12)NC=3N=CN=C4SC=CC43
Target:
CDK

References

Van Duyne R, et al. Effect of mimetic CDK9 inhibitors on HIV-1-activated transcription. J Mol Biol. 2013;425(4):812-829.